Fasoracetam (110958-19-5)

E se eka 7, 2021

Cofttek ke moetsi oa phofo ea Fasoracetam ho fetisisa China. Fektheri ea rona e na le sistimi e felletseng ea taolo ea tlhahiso (ISO9001 & ISO14001), e nang le tlhahiso ea khoeli le khoeli ea 150kg.

 


Boemo: Ka Phatlalatso ea Mesebetsi
Sehlopha: 1kg / mokotla, 25kg / Drum

Fasoracetam (110958-19-5) Slitšobotsi

Name: Fasoracetam
CAS: 110958-19-5
Ho hloeka 98%
Limolek'hule Mokgwa wa ho Nahana: C10H16N2O2
Boima ba limolek'hule: 196.250 g / mol
Melt Point: 57 ° C
Lebitso la k'hemik'hale (R) -1 - ((5-Oxo-2-pyrrolidinyl) carbonyl) piperidine
Li-synonyms: Fasoracetam; N- (5-Oxo-D-prolyl) piperidine; NS-105; NFC-1; LAM-105.
InChI Key: GOWRRBABHQUJMX-MRVPVSSYSA-N
Halofo ea bophelo: dihora tse 1.5
Solubility: Ho qhibiliha ho DMSO
Boemo ba ho Boloka: 0 - 4 C bakeng sa nako e khuts'oane (matsatsi ho isa ho libeke), kapa -20 C nako e telele (likhoeli)
e sebetsa joang: Fasoracetam ke sethethefatsi se bohlale kapa nootropic eo e leng ea lelapa le tummeng la li-racetam tsa lithethefatsi.
Ponahalo: Pula e tšoeu

 

Fasoracetam (110958-19-5) Ponahalo ea NMR

Fasoracetam (110958-19-5) - NMR Spectrum

Haeba o hloka COA, MSDS, HNMR bakeng sa sehlopha ka seng sa sehlahisoa le tlhaiso-leseling e ngoe, ka kopo ikopanye le rona mookameli oa papatso.

 

Fasoracetam ke eng (110958-19-5)?

Fasoracetam (110958-19-5) e tsejoang hape e le LAM-105, NFC-1, le NS-105, ke setlhare se bohlale kapa nootropic e leng ea lelapa le tummeng la li-racetam tsa lithethefatsi. Li-nootropics li hola ka potlako ho tsebahala ka lebaka la bokhoni ba tsona ba ho ntlafatsa ts'ebetso ea ts'ebetso, haholo-holo mesebetsi ea phethahatso, tšusumetso, mohopolo kapa boiqapelo ho batho ba phetseng hantle.

 

Fasoracetam (110958-19-5) melemo

Ts'ebetso e ntlafalitsoeng le tsepamiso

Fasoracetam e na le monyetla oa ho kenya tšebetsong maemo a Choline bokong, ho thusa basebelisi ho ikutloa ba tsepamisitse maikutlo hantle le ntlheng, ntle le tlhoko ea ho sebelisa tse ling tse khothatsang. Ho fapana le tse susumetsang, nootropic ena eu nolofalletsa ho lula u tsepamisitse maikutlo le ho etsa mesebetsi eohle e ka pele ho uena ntle le ho ikutloa eka o tsamaea hohle ho lokolla matla a mmele a ahileng. Ka mantsoe a bonolo, u tla ikutloa u khobile matšoafo 'me u lule u tsepamisitse maikutlo mosebetsing oa hau.

Ho eketseha ha likhahla tsa choline le hona ho ka lebisa ho khatello ea kelello e ntlafalitsoeng. Sena se bolela hore basebelisi ba sethethefatsi sena ba ka ba betere ha ba ithuta ba bile ba sebelisa bohlale ba bona maemong a nepahetseng.

Fasoracetam phofo ke sethethefatsi se hantle ho feta mang kapa mang ea batlang ho ntlafatsa mesebetsi ea bona ea kelello le ho fihlela litlatsetso tseo ba li hlokang, ntle le ho ikutloa a le sephara ebile a sa khone ho lula a khutsitse sebakeng se le seng.

Melemo ena ea Fasoracetam e boetse e nepahetse ho batho ba tsofetseng ba nang le ho fokotseha hoa kelello. Ka ho sebelisa fasoracetam, ba tla ba le bokhoni ba ho bua hantle, ba utloisise se etsahalang haufi le bona hape ba utloe ba le banyenyane ho latela monahano le kahlolo.

 

Ho fokotsa khatello ea maikutlo le matšoenyeho

Mofuta o mong oa phofo ea Fasoracetam (110958-19-5) o etsang hore o fapane le mofuta o fe kapa o fe oa matšoenyeho ke hore o fana ka phomolo e seng lemallo le e boreleli ho ts'oenyeha ntle le 'buzz' e amanang le eona. Meriana ena e etsa sena ka litlamorao tsa eona ho li-receptor tsa li-neurochemical tsa rona tse peli tse kholo tse susumetsang maikutlo tse leng glutamate le GABA.

Batho bao ba nang le matšoenyeho ba tloaetse ho ba le ts'ebetso e fetelletseng ea glutamate. Seo fasoracetam e se etsang ke ho lekanya tsamaiso eo. Hape, e hlohlelletsa li-receptor tsa GABA holimo, ka hona e fana ka khutso e sa tsamaelaneng le ho otsela.

Litlamorao tse ntle tsa phofo ea fasoracetam ha e felle feela ho batho. Setsebi se seng sa fasoracetam nootropics se boletse hore liphoofolo le tsona li bontšitse bokhoni ba ho sebetsana le maemo a thata ka khutso e kholo ka mor'a ho sebelisa moriana nakong ea liteko.

 

Fasoracetam (110958-19-5) sebelisa khanya?

Ntlafatso e ntlafetseng

Liphetoho tse fetolang maikutlo tsa fasoracetam ha li hang. E sebetsa ho tliseng motho boemong bo botle ba kelello butle-butle ha nako e ntse e tsamaea. Nako le nako ha mosebelisi a nka tlatsetso ea Fasoracetam, lithethefatsi li eketsa katleho ea li-receptor tsa GABA. Hopola hore ho netefalitsoe ka mokhoa oa bongaka hore boemo bo fokotsehileng ba ts'ebetso ho li-receptor tsa GABA bo ka baka mofuthu o mongata.

Ho nahanoa hore likarolo tse matlafatsang ts'ebetso ea GABA receptor e ka ba boselamose bo bocha ba likhomphutha tsa antidepressant tse nang le mefuta e mengata ea ts'ebeliso. Ke kahoo fasoracetam e ka sebetsang hantle bakeng sa basebelisi ba nang le maikutlo a tlase le boitšepo.

Haeba u ba le matšoenyeho sechabeng 'me u ikutloa u nyahame ka linako tsohle, fasoracetam e ka u thusa hore u ikutloe u le betere mme ea u isa boemong bo botle ba kelello le tšusumetso. Ho tsotehang le ho feta ke hore le ha o ka emisa ho e amohela, li-receptor tsa GABA li ntse li tla ntlafala mme o ke ke oa itšetleha ka meriana hore o hlaphoheloe.

 

Ho hopola mohopolo

Joalokaha re boletse pejana, Fasoracetam nootropic e sebetsa ka lik'hemik'hale tse seng li le teng bokong, tse kenyeletsang acetylcholine le choline, mme ka litlamorao tsena, e fana ka ts'ireletso e ntle ea ts'ireletso kahare ho boko ba rona. Ntle le moo, joalo ka li-Nootropics tsa lelapa la Racetam, e boetse e na le litšoaneleho tse ntlafatsang ho boloka mohopolo.

Ha u sebelisa meriana ena, u tla ba le mohopolo o molemohali oa ho hopola. Hape o tla ba le bokhoni ba ho theha mehopolo hantle. Se boleloang ke sena ke hore haeba u ithuta ho hong ha u ntse u le moriana ona, u tla ba le bokhoni ba ho boloka tsebo ena ka katleho. Ntle le moo, e thusa moloko oa khale ho loants'eng ho senyeha hoa memori ka mokhoa o nepahetseng mme e ba le mohopolo o motle ka ho feta ha ba ntse ba tsofala.

 

Fasoracetam (110958-19-5) tekanyo

Litlamorao tsa sethethefatsi sena ho batho ha li so ngolisoe ka botlalo, ka hona ha ho tataiso e hlakileng bakeng sa litekanyetso tsa fasoracetam.

Litekong tsa bongaka tse amang bacha ba nang le ADHD, fasoracetam e ne e fanoa ka molomo ka tekanyo e le 'ngoe ea 50 mg ho isa ho 800 mg, e lateloe ke litekanyo tse latelang tse tsamaisoang ke matšoao a fihlang ho 400 mg makhetlo a mabeli ka letsatsi libeke tse' ne. E mong oa fasoracetam psychonaut o nkile feela 10mg ka letsatsi ka mokhoa o nyane mme o atlehile ho fihlela litholoana tse lakatsehang.

Phuputsong ea bongaka e amang banna ba 14 ba Majapane, ho ile ha fanoa ka tekanyetso ea letsatsi le letsatsi ea 100 mg. Tekanyo ena e ipakile e sebetsa hantle. Leha ho le joalo, fasoracetam ke motsoako o matla haholo, 'me litekanyo tse tlase ho 20 mg tse tsamaisoang hanngoe kapa habeli ka letsatsi li ipakile li sebetsa ho basebelisi ba bang.

Ka li-Nootropics tsohle le ka fasoracetam, ho bohlale ho qala ka litekanyetso tse tlase tse sebetsang hantle mme butle-butle o eketsehe kamoo ho hlokehang.

 

Fasoracetam phofo Ho rekisoa(Moo u ka rekang phofo ea Fasoracetam ka bongata)

Khamphani ea rona e thabela likamano tsa nako e telele le bareki ba rona hobane re tsepamisa maikutlo mosebetsing oa bareki le ho fana ka lihlahisoa tse ntle. Haeba o rata sehlahisoa sa rona, re feto-fetoha le maemo ka mokhoa oo re ratang ho odara ka oona o lekanang tlhoko ea hau le nako ea hau ea kapele ea li-odara e tiisa hore o tla latsoa sehlahisoa sa rona ka nako. Re shebile hape le lits'ebeletso tse kenyellelitsoeng boleng. Re fumaneha bakeng sa lipotso tsa ts'ebeletso le tlhaiso-leseling ho ts'ehetsa khoebo ea hau.

Re mofani oa litsebi oa phofo ea Fasoracetam ka lilemo tse 'maloa, re fana ka lihlahisoa ka theko ea tlholisano,' me sehlahisoa sa rona ke sa boleng bo holimo haholo 'me se etsoa liteko tse thata, tse ikemetseng ho netefatsa hore se bolokehile hore se ka sebelisoa lefatšeng ka bophara.

 

References

[1] Ogasawara T, Itoh Y, Tamura M, le al. Ho kenyelletsoa ha litsamaiso tsa cholinergic le GABAergic ho khutliseng ts'oaetso ea memori ke NS-105, e matlafatsang tsebo. Pharmacol Biochem Behav. 1999; 64 (1): 41-52. doi: 10.1016 / s0091-3057 (99) 00108-2

[2] Elia, J., Ungal, G., Kao, C. le ba bang. Fasoracetam ho bacha ba nang le ADHD le glutamatergic gene network variants e sitisang mGluR neurotransmitter signaling. Nat Commun 9, 4 (2018).

[3] Foran E, Trotti D. Glutamate bapalami le tsela ea excitotoxic ea ho senyeha ha motor neuron ho amyotrophic lateral sclerosis. Pontšo ea Antioxid Redox. 2009; 11 (7): 1587-1602. doi: 10.1089 / ars.2009.2444